SARMs

Recently an absolutely new class of performance enhancing drugs was discovered. These drugs were called selective androgen receptor modulators (SARMs). Their initial purpose was increase of muscle mass in cancer patients, and they showed promising results, although not all of them passed through clinical trials.

Since their mass building and fat burning effect was comparable with steroids, they quickly became popular among bodybuilders. What is most important, they had no steroid-specific side effects, such as testicular atrophy, hepatotoxicity, growth of body hair etc.

Why SARMs are better than steroids

Steroids have two types of effect – anabolic and androgenic. Anabolic effect initiate protein synthesis inside muscle cells, which causes muscle growth and has fat burning effect. But
they also affect liver, heart, sex organs and secondary sexual characteristics (e.g. voice deepening, body hair growth, acne etc.). This is androgenic side of steroids.

If we regard testosterone as an example, its anabolic-to-androgenic ratio is 1:1. Meanwhile the anabolic-to-androgenic ratio of SARMs starts from 3:1 and goes up to 90:1. In other words SARMs can provide muscle gains and fat loss without the risks of gynecomastia and virilization.

Unlike most steroids, one can take SARMs orally, which is very convenient. Besides, you can buy SARMs legally. However, in case of changes in the law, SARMs producers and sellers protect themselves from legal issues with the label “for research purposes only” or “not for human use”.

Although there is a lot SARMs, here we will regard the most popular representatives of SARM family. Besides one should mention that most of them are on clinical or preclinical trial. Therefore, if you decided to use them, you do it at your own risk.

MK-2866

Ostarine SARM
Ostarine SARM

MK-2866 (aka Ostarine) induces muscle growth and has fat burning effect. It is probably one of the most studied SARMs. It passed through clinical trials and revealed great results without significant side effects.

During human trials aged men took MK-2866 for 3 months. As a result they gained 3 pounds of muscle mass and lost 1 pound of fat. What is more important, they had no changes in diet or exercises.
The similar results were obtained in cancer patients.

Side effects of MK-2866

These studies revealed no side effects. Nevertheless, there are reports that at high doses for long time (2-3 month) it may temporally suppress testosterone production. However, the levels of testosterone retuned to normal level in two weeks after drug discontinuation.

Doses of MK-2866

There are no official doses for SARMs usage. Therefore, we will regard the most “cautious” doses based on individual reports in forums.

The most optimal dose of Ostarine is 15-20 mg daily for 1 month. Then take a break for 1 month before a new cycle.

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LGD-4033

LGD-4033 (VK5211, Ligandrol)
LGD-4033 (VK5211, Ligandrol)

LGD-4033 (aka Ligandrol) went through multiple trials, and revealed very interesting resu lts: It greatly increased lean body mass in healthy men, who took this drug for 3 weeks. The result is dosage dependent, but even 1 mg is enough to accelerate muscle growth significantly.

Even at 22 mg daily it had no side effects or heath issues. In animal trials LGD-4033 showed great increase of bone density, muscle growth, and libido, without any adverse effect on prostate or liver. LGD-4033 has no fat burning effect. Therefore, during solo usage you will get more muscle mass but will not become leaner.

Side effects of LGD-4033

LGD-4033 can temporally suppress endogenous testosterone. However, it rather quickly returns to normal level after discontinuation of the drug (within 3 weeks).

That is to say if the level of your testosterone is low, you should be very careful while taking any SARM.

Doses of LGD-4033

At the dosage 2-5 mg daily for 1 month LGD-4033 will bring you very good results. As the result is dosage dependent, some bodybuilders take up to 15 mg/day. However, it is risky, since it may greatly suppress endogenous testosterone. Take 1 month break between cycles.

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GW 501516

GW 501516 (Сardarine)
GW 501516 (Сardarine)

GW501516 (aka Cardarine) have no official human trials. In mice it greatly increased endurance. For example during 4 weeks of GW501516 intake mice increased the running time by 68% and running distance by 70 %.

What is more important GW501516 caused growth of mitochondrial in muscle cells. It allows the muscles to produce more power and experience less fatigue. It also has fat burning properties which occur without destruction of muscle fibers. Thus with Cardarine you can improve endurance and get leaner without loss of muscles.

Side effects of GW501516

There are reports that GW501516 can cause cancer. However if we regard the study on which this rumor is based on, we will see that this statement is ridiculous. During this “carcinogenic” experiment mice were taking the human equivalent of 2400 mg a day for 2 years straight. That is 240 times more than the recommended dose, taken every day, for 2 years instead of 1 month!

There is not a single evidence that Cardarine can cause cancer at recommended doses. Besides there are no reports that it can suppress testosterone. Nevertheless, it does not mean that it has no side effects. This is a new drug, and we don’t know everything about it. Therefore, you should take it with caution.

Doses of GW501516

The optimal dosage of GW501516 is 10 mg / day. Divide the daily dosage into two portions. Take 5 mg in the morning and the other 5 in the afternoon. The duration of GW501516 cycle is 4 weeks, and then take 4 week pause before another cycle. You can also combine it with LGD-4033 and MK-2866.

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S4

S4 (aka Andarine) is probably one of the first SARMs which appeared in sports pharmacology. Athletes report moderate strength and muscle gain, and also fat loss. It’s better to combine Andarine with other SARMs, for example MK-2866 and LGD-4033.

Side effects of S4

There are report that S4 can cause visual abnormality, e.g. altered color perception or nighttime blindness. This is probably due to binding of its metabolite to receptor in the eyes. However this side–effect has no official confirmation.

Doses of S4

The optimal dosage is 50 mg daily. Divide it into two (25 mg) portions. Take it for 4 weeks, then make a 4 week gap and then repeat.

SR9009

SR9009 (Stenabolic) increases stamina endurance and produces fat burning effect. Besides it has anti-inflammatory effect and induces growth of new mitochondria in muscle cells.

The only disadvantage of this wonder drug is that it is injectable. Oral intake provides only 2% of bioavailability. However some manufacturers claim that you can take it orally, but it’s not the case

Conclusions

SARMs represent an excellent alternative to anabolic steroids (Testosterone etc.). Some of them are tested for a rather long time and have very good reputation among athletes, for example MK-2866, LGD-4033 и GW501516.

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Aromasin (Exemestane)

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ANTI-ESTROGEN
POST CYCLE THERAPY

Introduction

Exemestane (Aromasin) is a third generation aromatase inhibitor. In medical practice Exemestane is used as a treatment for breast cancer in postmenopausal women. In sports it is popular among athletes for its ability to suppress estrogenic side effects of AAS.

Its mechanism of action is similar to other aromatase inhibitors, such as Letrozole and Arimidex (Anastrozole). However, unlike them, athletes often use Exemestane after steroid cycle.

Since many AAS are prone to aromatization (i.e. conversion into female hormones) it leads to estrogen related side effects. They include water retention and gynecomastia. The latter is probably the worst of them. As to the water retention, it may significantly increase blood pressure.

One should remember that non-aromatizable steroids may also cause estrogenic side-effects if they have progestogenic activity. For instance, Nandrolone Decanoate has 5 times less aromatization in comparison with Testosterone. However, it may cause gynecomastia through progestogenic activity.

Exemestane is able to eliminate the risks of estrogenic side effects. According to the recent study, it reduces the levels of estradiol by 85 percent. Besides, when taking Aromasin (Exemestane) after steroid cycle one can speed up the secretion of endogenous testosterone.

Therefore some bodybuilders include Exemestane into PCT plan. Letrozole and Arimidex (Anastrozole) have similar effects. They send a signal to pituitary about the necessity for gonadotropic hormones (luteinizing and follicle-stimulating).

However, Exemestane has some advantages over these drugs

  • Has low androgenic activity.
  • Accelerates secretion of insulin-like growth factor

Effects

By using Exemestane after steroidcycle one can faster restore the endogenous testosterone production. Besides, it increases the levels of insulin-like growth factor, thus enhancing anabolism.
The effects of Exemestane

  • Prevents gynecomastia.
  • Suppresses the level of female hormones.
  • Increases anabolism
  • Improves muscular relief.
  • Prevents hypertension.
  • Reduces the negative effect of estrogens on HPTA.

It is important to know that only aromatizable and progestogenic steroids can cause estrogenic side-effects. The primary aromatizable steroid is Testosterone. However, its derivatives can enhance the work of estrogens, for instance methandienone.

Meanwhile the rate of aromatization of Boldenone Undecylenate is 50 percent in comparison with Testosterone. This is not enouph for a rapid increase of estrogen levels. Although Trenbolone and Nandrolone Decanoate have very low level of aromatization, their progestogenic activity may increase the concentration of female hormones to critical level.

The susceptibility to estrogenic (progestogenic) side-effects greatly depends on genetic predisposition of an athlete. However if you use these drugs in combination with easily aromatizing steroid, the risk of estrogenic side effects increases.

No matter what steroid you use, Exemestane will protect you from side effects. In sports pharmacology there are steroids based on dihydrotestosterone derivatives. Basically they are not aromatizable. An exception to this rule is oxymetholone, which has estrogenic activity.But it does not interact with aromatase, therefore Aromasin (Exemestane) will have no effect during Anapolone cycle.

Dosage and Usage

Now let’s regard the usage of Exemestaneafter steroid cycle. We know that AAS can suppress the endogenous testosterone production. The degree of this negative effect depends on the doses of steroid you use.

One should remember that even the lightest steroid at high doses can negatively affect HPTA. After steroid cycle the body begins to produce testosterone again, but only when exogenous hormone is over.
It takes a lot of time for the body to recover and it depends on the individual characteristics of an athlete’s organism. In worst case it takes about a year. The testosterone deficiency is abnormal for the body, and it may lead to definite health issues. For example is increases the levels of cortisol, which destroys muscles, and decreases sex drive.

Therefore, you should follow PCT (Post Cycle Therapy) in order to speed up testosterone production. Some bodybuilders take Aromasin during PCT in order to accelerate testosterone synthesis and increase the level of insulin-like growth factor. However, we do not recommend it, since the balance of female and male hormones is also important for the body.

Scientists found out that estradiol regulates the balance of lipoproteins, affects the libido etc. Thus by suppressing its production you can adversely affect other functions of your body. That’s why we recommend using Exemestane only during steroid cycle.

The recommended doses of Aromasin (Exemestane) vary from 12.5 to 25 mg every other day. However, in most cases it is enough for an athletes to use 12.5 mg no more than three times a week. If you take maximal doses, then the duration of Aromasin (Exemestane) cycle should not be long.

Use 25 milligrams only in the case of cholesteroldis balance. In other cases take minimal doses. Competitive bodybuilders also take Exemestaneone or two weeks before the contest in order to improve muscular relief.

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Testosterone Enanthate

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Testosterone Enanthate 250

General

"We are number one!" – this slogan the best suits to describe all testosterone-containing products. It’s virtually impossible to find serious bodybuilder, which does not use testosterone in his pre-season stacks. This is one of the best products for mass-gain. Great price/effect ratio makes testosterone unbeatable by other gear. It’s a king of all steroids.

Testosterone is the  major  and most important male androgen in the body, which carries many important functions, one of them is muscle growth. This makes testosterone the first steroid for bodybuilding. There is simply nothing more powerful. One may ask then – why other steroids still exist? The answer is that although testosterone is number one – it’s not ideal and still has certain disadvantages and different gear fill their own unique niches.

Testosterone enanthate as well as its close relative Testosteron Cypionate are long-acting esters. The main difference is molecular weight and size. Cypionate molecule is slightly heavier while still containing the same amount of active substance (testosterone). Therefore, let’s say 100 mg of testosterone enanthate contains ~12% more actual testosterone than 100 mg of cypionate (but less than for instance testosterone propionate or testosterone suspension). From the other hand, longer molecule takes more time to take apart thus making steroid more long acting. So, cypionate produces its effect for slightly longer time. But basically both steroids are almost the same.

Long-acting steroids require less injections (maybe 1 shot per week), so they are more convenient to use comparing to short-living ones like testosterone propionate or testosterone suspension, which contains 100% of testosterone per claimed concentration but also leaves body quickly and require injections every other day.

One should be aware that when you cease using long-acting gear its effects as well as side-effects still take place for 3-4 weeks, so short-living forms are easier to watch and control.

Testosterone aromatizes easily (i.e. part of it is being converted to estradiol). But more important point is that besides estrogen testosterone easily converts to dihydrotestosterone (DHT) thus increasing its androgenic properties (action on the prostate, body hair growth, increasing libido, unfortunately DHT is almost inactive in muscle cells).

According to scientific research, usage of high testosterone dosages increases the number of androgen receptors in muscle fibers. Another study shows that -I quote- Usage of anabolic steroids and particularly testosterone in combination with power training provokes an increase in muscle size as a result of their hypertrophy, and due to the formation of new muscle fibers. The key factor to this is the activation of muscle satellite cells, which increases substantially when taking large doses of steroids -end of quote-. Furthermore, it was also proven experimentally that usage of testosterone enanthate at a weekly dose of only 3 mg per kg of body weight raises growth hormone levels in the blood by 22% and insulin growth factor on 21%.

In simple words, when you take testosterone your existing muscle cells are growing by themselves and also they are producing new cells, which results in substantial muscle gains and increase in power. New muscle fibers normally appear when high dosages used. Besides this, there are also many other positive factors (general feeling of well-being, improved immune system, increased libido, etc.), as well as side effects, which we should consider.

Single purpose of testosterone enanthate is a help in mass-gain. Aromatization (conversion to estrogen) plays here some positive role. Testosterone-Enanathate has great effect on both – novices and advanced users.

The effectiveness of testosterone depends on the amount of certain enzymes in the body. For testosterone, as well as for nandrolone, a "critical" enzyme is a 5-Alpha-Reductase. Especially important this enzyme is for long-acting esters of both steroids. The increased amount of 5-Alpha-Reductase leads to accelerated conversion of testosterone to dihydrotestosterone (DHT). The latter is good for increasing libido, but not to build muscle. As you recall, in muscle fibers DHT is practically inactive (unlike in the skin and prostate). In addition, DHT is not so bad as anti-estrogen, but at high level this is not good for muscle gains (on one hand you try to kill estrogen to avoid side effects, on other hhand, estrogen helps to build muscle size). Therefore, testosterone and nandrolone are not ideal agents for athletes with elevated level of 5-Alpha-Reductase enzymes. How to find out your 5-Alpha-Reductase level? Either by taking special medical tests or by carefully watching your body reaction on different steroids

Dosage and usage

Inject every 5-7 days (more frequent shots will slightly increase the effect) , preferably into big muscles like upper leg or buttocks. Rotate injection spots to prevent inflammation.

Some PROfessional bodybuilders and powerlifters do 2000mg (2 grams) of testosterone enanthate daily. But such people do not need our advice and we don’t think this is a good idea for everybody. Most of advanced users will be very happy with a dosage 2000 mg / week if used standalone. Novices can do 500 mg/week, effect from lower dosages is not that notable. If you do below 500 mg stacking with anabolic substances like deca is necessary. 250 mg/week is the lowest possible volume, but better stay with 500 mg / week.

Stacking

Testosterone is very powerful substance by itself to allow standalone cycles. So 500-1000mg of testosterone enanthate or cypionate (both are long-acting) will produce notable results over 8 or better 10 weeks cycle whether used in combo or standalone. 12 week stacks also often takes place since this product is non-toxic. Testosterone has so many different activities that other steroids serves merely as an additional supplement. However, stacking is necessary if athlete have serious goals. It helps to reduce the quantity of testosterone and thus negative side effects by adding some milder substances like Primobolan Depot (Methenolone Enanthate), Nandrolone Decanoate (Deca-Durabolin) or Boldabol (Equipoise).

Testosterone is in fact an ideal partner for any other steroid because of its action on androgen receptor in muscle cells and it’s possible to combine it virtually with everything. The best results, however, are achieved when testosterone enanthate is combined with Nandrolone Decanoate esters, Methandrosterolone or Anadrol/Anapolon (Oxymetholone). Combination of testosterone enanthate + Nandrolone Phenilpropionate + Methandrosterolone provides bulking "super action". Stacking of testosterone enanthate with Trenbolone or Boldabol (Equipoise) produces great results as well.

Common length of testosterone enanthate cycles is 8-10 weeks, sometimes 12 weeks.

A popular "mass" stack is 500 mg of testosterone enanthate / week + 400 mg of Nandrolone Decanoate (Deca-Durabolin) / week and strong PCT – you need anti-estrogen during and after cycle and you need to boost natural production afterwards.

For those who are looking for milder bulking stack – the same testosterone dosage in combination with primobolan 400-600 mg/week is an option. It makes cycle much safer although gains will be also lower because primobolan has lower anabolic properties comparing to deca, it’s main advantage is non-aromatization. As we already mentioned low estrogen level leads to lower mass gains although the gains you receive will be more lean and dry. Another disadvantage is high price of Primobolan. PCT and anti-estrogen are still needed as always with testosterone.

Third option is testosterone enanthate with Boldabol (Equipoise) 200-400 mg/week, which is stronger than deca (nandrolone) and has lower side-effects. This is still bulking stack, however, boldenone provides more lean and dry mass gains, which is similar to positive effects of primobolan, although much stronger. Furthermore, boldenone promotes appetite, which is often suppressed by usage of testosterone thus making your nutrition more effective.

As it was mentioned before, you can stack testosterone virtually with everything, but nandrolone, primobolan and boldenone are the best options for bulking cycles. As for other gear – you should consider what kind of effect they can add. For instance oxandrolone (anavar) will add some strength and might be used in pre-competition cycle when bulking is not necessary. If you are looking only for mass – you may simply increase testosterone dosages and no need to add other compound UNTIL side effects will prevail. Only after this it worth stacking (or if you are looking for milder cycle from the beginning). To explain this thought read following example. For instance, someone wants purely bulking cycle. He tried once, did 250 mg/week and was not satisfied with the results. What to do next time? Not ideal decision would be 250 mg of test in combo with 400 mg of deca. Ideal and simple decision 500 mg of testosterone /week. Another example, someone is looking for a moderate bulking cycle. Not too weak, not with a lot of side effects as well but rather something on the middle. A possible solution is 250 mg of testosterone/week and 200 mg of boldenone/week with PCT, of course. Hopefully you understood what author means.

Some other cycle examples

Nomal cycle:
500 mg testosterone enanthate/week +
Turanabol (Turinabol) or Anavar (Oxandrolone) 40-50 mg / day

Pre-competition cycle for advanced users, 8 weeks. Start with testosterone enanthate and testosterone cypionate 400 mg/week each, decrease smoothly to 100 mg on the last week. At the same time do Anavar (Oxandrolone) starting from 80 mg / day and decrease by 10 mg every week until you reach 10 mg/day on the last week. For amateur users dosages of testosterone starts 200 mg/week and fall down to 25 mg/w on the last week with the same dosage of anavar, although on my opinion this is extreme case.

"Super" stack for PRO:
Anadrol/Anapolon (Oxymetholone) 100-150 mg / ED for 8 weeks +
Nandrolone Decanoate (Deca-Durabolin) 400 mg/week for 7 weeks, decrease dosage on last two weeks +
Testosterone Enanthate 500-1000 mg (peak on the mid) for 10 weeks +
Testosterone Cypionate 400-800 mg / week (peak on the mid) +
Dianabol 50-20 mg on weeks 8-11.

Anti-estrogen is needed starting from week 2 or 3 till the end and HCG is needed on weeks 4-5 and 9-11, 5000 IU / week. Tamoxifen/Clomiphen is still needed after the cycle to boost natural hormone production, HCG will just smoothen this downfall.

Detection times

It has long detection time as most of testosterones, especially long-acting ones. Doping tests can find it up to three months after the cycle.

Side effects and PCT (Post Cycle Therapy) with testosterone Enanthate

Since testosterone is easily aromatized, its use in high doses may cause side effects such as water retention, acne, female-pattern fat deposits, and gynecomastia ("bitchy tits"). But for most athletes these problems start at high doses of the drug – from 1 gram (1000mg) per week or more. Therefore, it is advised to take some anti-estrogen like Arimidex (Anastrozole), Proviron (Masterlone), Tamoxifen (Nolvadex) or Clomiphene (Clomid). At dosages of 500-600 mg per week, side effects are normally low, but some people are more prone (more sensitive) to these side effects than others, so if problems arise, do 1 tab of :clomiphen: 50mg or tamoxifen 20mg until problem disappear.

The conversion of testosterone to DHT means a risk of such androgen-related side effects as baldness and prostate enlargement. Again, this only applies to high dosages or to the people with high level of 5-alpha-reductase enzyme.

The use of testosterone, even at doses of more than two grams (2000mg) a week not infringe either the liver or other organs. Recovery of natural testosterone production after a cycle is normally quick and successful.

PCT: 25-50mg of arimidex / day OR 25-50 mg of proviron / day during the cycle. Normally 25 mg is just fine but in case of "heavy" cycles dosages up to 100 mg of proviron might be required. Actually, it’s better to use Proviron (Masterlone) instead of Arimidex (Anastrozole) along with the testosterone injections since it increases volume of free testosterone in the blood thus promoting gains. Athlete should also consider the following thing – estrogen converted from androgen plays very important role in muscle gains. Thus, more anti-estrogen you use – there are less estrogen-related side effects but also less gains. So, you have to find experimentally what suits the best to your body. People who worry more about gains should use minimal dosage of anti-estrogen, people who worry more about estrogen level should use higher one.

Some people are more concerned about androgen-related side effects such as deep voice, baldness, prostate hypertrophy. These ones should do 1 tab / ED of a product named finasteride (brand names propecia, proscar, fincar, etc.), which blocks 5-alpha-reductaze and thus conversion of testosterone into more aggressive androgenic substance DHT. Again, one should find a balance. DHT is more powerful androgen, maybe 300% stronger than testosterone and it’s positive effects increases along with unwanted side effects. Also, keep in mind that if you are more concerned about androgen-related side effects, you should not use Proviron, which is in fact very similar to :DHT:. Better use Arimidex (Anastrozole) as anti-estrogen in that case.

As you may see, all these things – testosterone, dihydrotestosterone, estrogen and androgen levels, estrogen blockers, etc. are highly related and dependant on each other so there is no single advice for everyone, you should consider what is more important exactly for you and choose appropriate anti-estrogen and dosage basing on it.

When the cycle is over, natural testosterone production is severely suppressed and needs to be restored, otherwise much of gains will be lost and also you’ll have problems with libido and shrinkage of testicles, which is especially true for long cycles. Many bodybuilders of 70es, when steroid science was not so developed felt all these side effects and became big and fatty or small and tiny or had heart problems (heart is also a muscle) which leaded to all these horror stories and prohibition of steroids in many countries. Fortunately, now we all know how to make it safe. Using Human Chorionic Gonadtropin (HCG, Pregnyl) and Tamoxifen (Nolvadex) (nolvadex, cymoplex, cytotam) / Clomiphene (Clomid) (clomid, fertomid) plays key role in Post Cycle Therapy. Let’s say 40 mg (2 tabs 20 mg) of Tamoxifen equals 150 mg (3 tabs 50 mg) of Clomiphene). People still argue, what is more effective. Many people believe tamoxifen is better during cycle and Clomiphene (Clomid) is better after it. However, there are also opposite opinions, so if you are in doubts combine tamo+clom during PCT after the cycle is over.

One should start HCG injections on the last week of cycle and do 1500-3000 IU every 5-7 days depending on testosterone dosages during the cycle. HCG serves as an alternative to natural LH, it will boost testosterone production in the body thus restoring size of testicles back to normal. HCG should be used for 2-4 weeks in total. However, it does not eliminate the problem but serves just as a "bridge" between the cycle and post-cycle healers – Tamoxifen (Nolvadex)/Clomid. Although it "orders" to the body to start producing testosterone, this is not "natural" production. In fact it even suppresses natural production of the hormone, and usage of HCG should be stopped two weeks before you finish Tamoxifen (Nolvadex) / Clomiphene (Clomid).

Using HCG is strictly advisable, but if you don’t have it, just start with higher then described below clomiphene/tamoxifene dosages, let’s say 3-4 tabs/ED for two weeks.

Two weeks after the cycle (if HCG has been used) start doing 2 tabs of tamoxifen 20 mg or 3 tabs of clomiphene 50 mg or combination of both for two weeks. After this, do two more weeks with 1 tab of tamoxifen or two tabs of clomiphene daily.

A conclusion: Arimidex or Proviron fight estrogen during cycle, tamoxifen and clomid finish this job and also boost natural testosterone production. HCG helps to smoothen critical testosterone production downfall right after the cycle.

Female usage

Amazingly, in medical practice testosterone enanthate is widely used in treatment of females and even children with certain pathologies. The only common thing between all these people is low testosterone level in the blood.

But it is strictly not advisable for females with normal testosterone level to use testosterone injections for sport-related purposes. External testosterone will simply lead to virilization effects, so women in bodybuilding should stay away from it. There are different ethers like testosterone undecanoate, which fit well for them.

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Efedrin [Ephedrine HCL]

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Ephedrine

Usage and stacking

For weight loss purposes especially effective in combination with caffeine and aspirin (salicin acid). Average daily dosage is 50 mg (split on two). Throw in 150mg of aspirin too. This will not only boost the effectiveness but also keep your blood pressure down and ensure your blood capillaries in your brain don’t go pop under the force.

!!! Taking ephedrine shouldn’t become a regular just an every so often thing or you will become de-sensitised to them and might get sick dependance.

Description

Ephedrine is a sympathomimetic amine – that is, its principal mechanism of action relies on its direct and indirect actions on the adrenergic receptor system, which is part of the sympathetic nervous system or SNS. Central nervous system or CNS involvement is present, but the predominant clinical effects are caused by involvement with the sympathetic segment of the peripheral nervous system. Due to the fact that while ephedrine does cross the blood-brain barrier, it doesn’t do this very efficiently (efficient crossers with similar modes of action would include amphetamine and methamphetamine).

Ephedrine increases post-synaptic noradrenergic receptor activity by (weakly) directly activating post-synaptic α-receptors and β-receptors, but the bulk of its effect comes from the pre-synaptic neuron being unable to distinguish between real adrenaline or noradrenaline from ephedrine. The ephedrine, mixed with noradrenaline, is transported through the noradrenaline reuptake complex and packaged (along with real noradrenaline) into vesicles that reside at the terminal button of a nerve cell.

As an alkaloid, having some small amount of ephedrine within a noradrenaline vesicle increases the overall pH of the vesicle. This has the effect of increasing likelihood that the affected vesicle will be released during any subsequent action potential the nerve cell experiences. The nerve cells in question generally fire at some regular baseline rate; the effect of adding ephedrine is to increase the number of vesicles released during each action potential and possibly to extend the time during which noradrenaline has an opportunity to have an effect on the post-synaptic neuron by virtue of the fact that the reuptake complex has to process both noradrenaline AND ephedrine, presumably a longer process.

Ephedrine’s mechanism of action on neurotransmission in the brain is wide. Its action as an agonist at most major noradrenaline receptors and its ability to increase the release of both dopamine and to a lesser extent, serotonin by the same mechanism as explained above for norepinephrine, is presumed to have a major role in its mechanism of action.

Because of ephedrine’s ability to potentiate dopamine neurotransmission it is thought to have addictive properties by some researchers. The ability to potentiate serotonin and noradrenergic activity is clinically relevant, but is not thought to contribute to the potential for abuse.

While ephedrine’s role in the serotonin system is less understood there is preliminary documentation of clinically significant agonism at excitory serotonin receptors, perhaps as a downstream response to the large release of norepinephrine in the nucleus accumbens (commonly referred to as the “pleasure center” of the brain). In mice, stereotypical behaviour was both easily induced by administration of ephedrine and its primary alkaloids and reversed when serotonin antagonists were administered.

Adverse effects

The approved maximum daily dosage of ephedrine for use as a bronchodilator is 150mg, as specified on the packaging of the bronchodilator and expectorant combination, Bronkaid, made by Bayer pharmaceuticals.

Overdose can lead to death, although the approved dose is not likely to cause severe reactions when used as directed.

Ephedrine can also lead to damage of the brain receptors’ over a period of high usage; this is because of its constant action on the neurochemicals. It also leads to high increase in blood pressure which over time can lead to damage in the blood vessels.

Contraindications

Ephedrine should not be used in conjunction with certain antidepressants, namely SNRIs (serotonin-norepinephrine re-uptake inhibitors), as this increases the risk of the above symptoms due to excessive serum levels of norepinephrine.

Bupropion is an example of an antidepressant with an amphetamine-like structure similar to ephedrine, and it is known as an NDRI (norepinephrine-dopamine re-uptake inhibitor). It has an action which bears more resemblance to amphetamine than to fluoxetine in that its primary mode of therapeutic action involves norepinephrine and to a lesser degree dopamine. But it also releases some serotonin from presynaptic clefts. It should not be used with ephedrine as it may increase the likelihood of the above side effects.

Ephedrine should be used with caution in patients with

  • inadequate fluid replacement
  • impaired adrenal function
  • hypoxia
  • hypercapnia
  • acidosis
  • hypertension
  • hyperthyroidism
  • prostatic hypertrophy
  • diabetes mellitus
  • cardiovascular disease
  • during delivery if maternal BP > 130/80 mmHg
  • and lactation

Contraindications for the use of ephedrine include: closed angle glaucoma, phaeochromocytoma, asymmetric septal hypertrophy (idiopathic hypertrophic subaortic stenosis), concomitant or recent (previous 14 days) monoamine oxidase inhibitor (MAOI) therapy, general anaesthesia with halogenated hydrocarbons (particularly cyclopropane or halothane), tachyarrhythmias or ventricular fibrillation, hypersensitivity to ephedrine or other stimulants. Ephedrine should NOT be used at any time during pregnancy unless specifically indicated by a qualified physician and ONLY when other options are unavailable.

It is common for many athletes to use stimulants while exercising. Such use of ephedrine has been associated with stimulant dependence, as well as deaths from heatstroke in athletes and circulatory problems such as aortic aneurysm in weightlifters, though these side effects are rare.

Ephedrine has been reported to cause both physical and psychological dependence after excessive long-term use. This is particularly true with oral forms of ephedrine, since parenteral administration is unlikely to occur over long periods.

A pity – not available now.

 

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Saizen – HGH (Somatropin)

Buy Jintropin - HgH
Merck Serono (Germany)
10 X 100 IU in amp & 10 X 1ml amp of water solution

Saizen (HGH, Human Growth Hormone) [Somatropin]

Saizen click.easy, is a recombinant human growth hormone (rHGH) for injection. It is a liquid consisting of the identical sequence of 191 amino acids of human growth hormone. The molecular formula is C990H1528N262O300S7. Its molecular weight is 22,125 Daltons.

As with no other doping drug, growth hormones are still surrounded by an aura of mystery. Some call it a wonder drug which causes gigantic strength and muscle gains in the shortest time. Others consider it completely useless in improving sports performance and argue that it only promotes the growth process in children with an early stunting of growth. Some are of the opinion that growth hormones in adults cause severe bone deformities in the form of overgrowth of the lowerjaw and extremities. And, generally speaking, which growth hormones should one take the human form, the synthetically manufactured version, recombined or genetically produced form and in which dosage? All this controversy about growth hormones is so complex that the reader must have some basic information in order to understand them.

The growth hormones is a polypeptide hormone consisting of 191 amino acids. In humans it is produced in the hypophysis and released if there are the right stimuli (e.g. training, sleep, stress, low blood sugar level). It is now important to understand that the freed HGH (human growth hormones) itself has no direct effect but only stimulates the liver to produce and release insulin-like growth factors and somatomedins. These growth factors are then the ones that cause various effects on the body. The problem, however, is that the liver is only capable of producing a limited amount of these substances so that the effect is limited. If growth hormones are injected they only stimulate the liver to produce and release these substances and thus, as already mentioned, have no direct effect.

The use of these STH (somatotropic hormone) compounds offers the athlete three performance-enhancing effects. STH has a strong anabolic effect and causes an increased protein synthesis which manifests itself in a muscular hypertrophy (enlargement of muscle cells) and in a muscular hyperplasia (increase of muscle cells.) The latter is very interesting since this increase cannot be obtained by the intake of steroids. This is probably also the reason why STH is called the strongest anabolic hormone. The second effect of STH is its pronounced influence on the burning of fat. It turns more body fat into energy leading to a drastic reduction in fat or allowing the athlete to increase his caloric intake. Third, and often overlooked, is the fact that STH strengthens the connective tissue, tendons, and cartilages which could be one of the main reasons for the significant increase in strength experienced by many athletes. Several bodybuilders and powerlifters report that through the simultaneous intake with steroids STH protects the athlete from injuries while inereasing his strength.

You will say that this sounds just wonderful. What is the problem, however since there are still some who argue that STH offers nothing to athletes? There are, by all means, several athletes who have tried STH and who were sadly disappointed by its results. However, as with many things in life, there is a logical explanation or perhaps even more than one:
1. The athlete simply has not taken a sufficient amount of STH regularly and over a long enough period of time. STH is a very expensive compound and an effective dosage is unaffordable by most people.

2. When using STH the body also needs more thyroid hormones, insulin, corticosteroids, gonadotropins, estrogens and what a surprise androgens and anabolics. This is also the reason why STH, when taken alone, is considerably less effective and can only reach its optimum effect by the additive intake of steroids, thyorid hormones, and insulin, in particular. But we must point out in this case that STH has a predominantly anabolic effect. There are three hormones which are needed at the same time in order to allow for maximum anabolic effect. These are STH, insulin, and an LT-3 thyroid hormone, such as, for example, Cytomel T3. Only then can the liver produce and release an optimal amount of somatomedin and insulin-like growth factors. This anabolic effect can be further enhanced by taking a substance with an anticatabolic effect. These substances are-everybody should probably know by now-anabolic/androgenic steroids or Clenbuterol. Then a synergetic effect takes place.`Are you still wondering why pro bodybuilders are so incredibly massive but, at the same time, totally ripped while you are not. Most athletes have tried STH during preparation for a competition in that phase when the diet is calorie-reduced.

The body usually reacts by reducing the release of insulin and of the L-T3 thyroid hormone. And, as was described under point 2, this is not an advantageous condition when STH is expected to work well. Well, we almost forgot. Those who combine Clenbuterol with STH, should know that Clenbuterol (like Ephedrine) reduces the body`s own release of insulin and L-T3. True, this seems a little complicated and when reading it for the first time it might be a little confusing; however it really is true: STH has a significant influence on several hormones in the human body; this does not allow for a simple administration schedule.

As said, :ST: is not cheap and those who intend to use it should know a little more about it. If you only want to burn fat with STH you will only have to remember user information for the part with the L-T3 thyroid hormone as is printed by Kabi Pharmacia GmbH for their compound Genotropin:

“The need of the thyroid hormone often inereases during treatment with growth hormones.”

3. Since most athletes vho want to use STH can only obtain it if prescribed by a physician, the only supply source remains the black market. And this is certainly another reason why some athletes might not have been very happy with the effect of the purchased compound. How could he, if cheap HCG was passed off as expensive STH?

Since both compounds are available as dry substances, all that would be needed is a new label of Serono`s Saizen or Lilly`s Humatrope on the HCG ampule. It is no longer fun when somebody is paying $200 for 5000 I.U. of HCG, only worth $ 12, and thinking that he just purchased 4 I.U. of STH. And if you think this happens only to novices and to the ignorant, ask Ben Johnson. “Big Ben,” who during three tests within five days showed an above-limit testosterone level, was not a victim of his own stupidity but more likely the victim of fraud. According to statistics by the German Drug Administration, 42% of the HGH vials confiscated on the North American black market are fakes. In addition to a display of labels in the Dutch or Russian language the fakes are distinguished from the original product, in sofar as the dry substance is not present as lyophilic but present as loose powder. The fakes confiscated so far use the name “Humatrope 16” under the name of Lilly Company (with Dutch denomination) or “Somatogen” (in Russian).” Nowhere can this much money be made except by faking STH. Who has ever held original growth hormones in his hand and known how they should look?

4. In a few very rare cases the body reacts by developing antibodies to the exogenous STH, thus making it ineffective. The question of the right dosage, as well as the type and duration of application, is very difficult to answer. Since there is no scientificresearch showing how STH should be taken for performance improvement, we can only rely on empirical data, that is experimental values. The respective manufacturers indicate that in cases of hypophysially stunted growth due to lacking or insuffieient release of growth hormones by the hypophysis, a weekly average dose of 0.3 I.U/ week per pound of body weight should be taken. An athlete weighting 200 pounds, therefore, would have to inject 60 I.U. weekly. The dosage would be divided into three intramuscular injections of 20 I.U. each. Subcutaneous injections (under the skin) are another form of intake which, however would have to be injected daily, usually 8 I.U. per day. Top athletes usually inject 4-16 I.U./day. Ordinarily, daily subcutaneous injections are preferred. Since STH has a half life time of less than one hour, it is not surprising that some athletes divide their dail dose into three or four subcutaneous injections of 2-4 I.U. each.

Application of regular small dosages seems to bring the most effective results. This also has its reasons: When STH is injected, serum concentration in the blood rises quickly, meaning that the effect is almost immediate. As we know, STH stimulates the liver to produce and release somatomedins and insulin like growth factors which in turn effect the desired results in the body. Since the liver can only produce a limited amount of these substances, we doubt that larger STH injections will induce the liver to produce instantaneously a larger quantity of somatomedins and insulin-like growth factors. It seems more likely that the liver will react more favorably to smaller dosages. If the STH solution is injected subcutaneously several consecutive times at the same point of injection, a loss of fat tissue is possible.

Therefore, the point of injection, or even better, the entire sisde of the body should be continuously, changed in order to avoid a loss of local fat tissue (lipoathrophy) in the injection cell. One thing has manifested itself over the years: The effect of STH is dosage-dependent. This means either invest a lot of money and do it right or do not even begin. Half-hearted attempts are condemned to failure Minimum effective dosages seem to start at 4 I.U. per day. For comparison: the hypophysis of a healthy; adult, releases 0.5-1.5 I.U. growth hormones daily.

The duration of intake usually depends on the athlete`s financial resources. Our experience is that STH is taken over a prolonged period, from at least six weeks to several months. It is interesting to note that the effect of STH does not stop after a few weeks; this usually allows for continued improvements at a steady dosage. Bodybuilders who have had positive results with STH have reported that the build-up strength and, in particular, the newly-gained muscle system were essentially maintained after discontinuance of the product. It remains to be clarified what happens with the insulin and LT-3 thyroid hormone.

Athletes who take STH in their build-up phase usually do not need exogenous insulin. It is recommended, in this case, that the athlete eats a complete meal every three hours, resulting in 6-7 meals day. This causes the body to continuously release insulin so that the blood sugar level does not fall too low. The use of LT-3 thyroid hormones, in this phase, is carried out reluctantly by athletes. In any case, you must have a physician check the thyroid hormone level during the intake of STH. Simultaneous use of anabolic /androgenic steroids and/or Clenbuterol is usually appropriate. During the preparation for a competition the use of thyroid hormones steadily inereases. Sometimes insulin is taken together with STH, as well as with steroids and Clenbuterol.

Apart from the high damage potential that exogenous insulin can have in non-diabetics, incorrect use will simply and plainly make you “FAT! Too much insulin activates certain enzymes which convert glucose into glycerol and finally into triglyceride. Too little insulin, especially during a diet, reduces the anabolic effect of STH. The solution to this dilemma? Visiting a qualified physician who advises the athlete during this undertaking and who, in the event of exogenous insulin supply, checks the blood sugar level and urine periodically.

According to what we have heard so far, athletes usually inject intermediately-effective insulin having a maximum duration of effect of 24 hours once a day. Human insulin such as Depot-H-Insulin Hoechst is generally used. Briefly-effective insulin with a maximum duration of effect of eight hours is rarely used by athletes. Again a human insulin such as H-Insulin Hoechst is preferred. The undesired effect of growth hormones, the so-called side effects, are also a very interesting and hotly-discussed issue. Above all it must be said: STH has none of the typical side effects of anabolic/androgenic steroids including reduced endogenous testosterone production, acne, hair loss, aggressiveness, elevated estrogen level, virilization symptoms in women, and increased water and salt retention.

The main side effects that are possible with STH are an abnormally small concentration of glucose in the blood (hypoglycemia) and an inadequate thyroid function. In some cases antibodies against growth hormones are developed but are clinically irrelevant. What about the horror stories about acromegaly, bone deformation, heart enlargement, organ conditions, gigantism, and early death? In order to answer this question a clear differentiation must be made between humans before and after puberty. The growth plates in a person continue to grow in length until puberty.

After puberty neither an endogenous hypersection of growth hormones nor an excessive exogenous supply of STH can cause additional growth in the length of the bones. Abnormal size (gigantism) initially goes hand in hand with remarkable body strength and muscular hardness in the afflicted; later, if left untreated, it ends in weakness and death. Again, this is only possible in pre-pubescent humans who also suffer from an inadequate gonadal function (hypogonadism). Humans who suffer from an endogenous hypersecrehon after puberty and whose normal growth is completed can also suffer from acromegaly. Bones become wider but not longer. There is a progressive growth in the hands and feet and enlargement of features due to the growth of the lower jaw and nose. What the authorities like to do now is to present extreme cases of athletes suffering from these malfunctions in order to discourage others and to drum into athletes the fact that with the exogenous supply of growth hormones they would suffer the same destiny. This, however, is very unlikely, as reality has proven.

Among the numerous athletes using STH comparatively few are seven feet tall Neanderthalers with a protruded lower jaw, deformed skull, claw like hands, thick lips, and prominent bone plates who walk around in size 25 shoes. In order to avoid any misunderstandings, we do not want to disguise the possible risks of exogenous STH use in adults and healthy humans, but one should at least try to be openminded. Acromegaly, diabpetes, thyroid insuficiency, heart muscle hypertrophy, high blood ressure, and enlargement of the kidneys are theoretically possible if STH is used excessively over prolonged periods of time; however, in reality and particularly when it comes to the external attributes, these are rarely present.

Some athletes report headaches, nausea, vomiting, and visual disturbances during the first weeks of intake. These symptoms disappear in most cases even with continued intake.

The most common problems with STH occur when the athlete intends to inject insulin in addition to STH. The substance somatropin is available as a dried powder and before injecting it must be mixed with the enclosed solution-containing ampule. The ready solution must be injected immediately or stored in the refrigerator for up to 24 hours. It is usually recommended that the compound be stored in the refrigerator. With the exception of the remedy Saizen the biological activity of growth hormones is usually not impaired when storing the dry substance at 15-25 C (room temperature); however, a cooler place (2-8° C) is preferable.On the black market the price for 4 I.U. each of the compounds Genotropin, Humatrope, Norditropin, and Saizen, in Europpe is $80-120 for a prick-through vial including the solution ampule. As already mentioned, there are many fakes. It is noted that for the U.S.-American growth hormones compounds, the substance content is not given in I.U.(International Units) but in mg (milligrams).

Since l mg corresponds to exactly 2.7 I.U. the 5mg solution of the compound Humatrope by Lilly contains exactl 13.5 I.U. of Somatropin. The 10 mg solution of the Protropin compound by the Genentech therefore contains 27 I.U. of Somatropin.

In American powerlifting and bodybuilding circles Humatrope is usually preferred over Protropin. The reason is that Humatrope is synthesized from a chain of 191 amino acids and thus is identical to the amino acid sequence of the human growth hormones. Protropin, on the other hand, consists of 192 amino acids, one amino acid too many. This might be the explanation for why more antibodies are developed with Protropin than with Humatrope. growth hormones are on the doping list but they are not yet detectable during doping tests.

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Zymoplex

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30 Tabs x 20mg Total 600mg

Zymoplex in bodybuilding (Tamoxifen Citrate, Nolvadex)

Nolvadex (Tamoxifen) belongs to a category and class of drugs known as selective Estrogen receptor modulators (SERMs). Selective Estrogen receptor modulators belong to an even broader class of drugs known as anti-estrogens. The other subcategory of drug under the anti-estrogens category is known as aromatase inhibitors (AIs), such as Aromasin (Exemestane) and Arimidex (Anastrozole). AIs and SERMs make up anti-estrogens. Aromatase inhibitors differ greatly from SERMs in their action and how they deal with the issues of estrogen control.

This drug is a potent nonsteroidal anti-estrogen. It is indicated for use in estrogen dependent tumors, i.e. breast cancer. Steroid users take Nolvadex to prevent the effects of estrogen in the body. This estrogen is most often the result of aromatizing steroids.

Nolvadex can aid in preventing edema, gynecomastia, and female pattern fat distribution, all of which might occur when a man’s estrogen levels are too high. Also, these effects can occur when androgen levels are too low, making estrogen the predominant hormone. This can occur when endogenous androgens have been suppressed by the prolonged use of exogenous steroids.

Nolvadex works by competitively binding to target estrogen sites like those at the breast. This drug is not toxic nor have any side effects been seen in athletes who used the drug’ as an anti-estrogen. This drug is the most popular anti- estrogen amongst steroid users. Although it does not turn out to be 100% effective for everyone, it does seem to exhibit some level of effectiveness for the majority.

Zymoplex in bodybuilding works so well for some bodybuilders they can take drugs like Anadrol right up to a contest as long as they stack it with Nolvadex. It would seem wise to take this drug in conjunction with any steroid cycle. Most reported a dosage of 10 mg to 20 mg daily got the job done.

Dose of Zymoplex (Tamoxifen Citrate, Nolvadex)

Dosage of Zymoplex (Tamoxifen Citrate, Nolvadex) is prescribed by health providers particularly. The main condition that influences on dose is the disease of the patient. If patients have breast cancer or kidney cancer, they must take 20-40 mg of Zymoplex (Tamoxifen Citrate, Nolvadex) 1-2 times daily (in the morning and in the evening). Persons that suffer of endometrial cancer usually take 20-30 mg of this drug 1-2 times per day. Tablets of this drug must be swallowed with a glass of water. They must not be chewed. Daily quantity is taken at once in the morning or it’s divided in 2 and it’s applied in the morning and in the evening. Duration of therapy with Zymoplex (Tamoxifen Citrate, Nolvadex) lasts usually long period of time. Benefits can be reached, if this drug is administrated needed time continually. Sometimes treatment with this medicine is combined with beam or cytostatic therapy.

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Zydena

Buy Zydena (Udenafil) online, Dong-A Pharmaceutical Co., Korea

Dong-A Pharmaceutical Co. (Korea)
4 Tabs x 100mg Total 400mg

Zydena (Udenafil)

Active Ingredient: Udenafil

Udenafil– trade name «Zydena ®» is one of the four molecules investigated for the treatment of erectile dysfunction with proven clinical efficacy, high safety and acceptability to the patient. The unique qualities of Zydena distinguish it from commercially available inhibitors of other members of the group focfodiesterazy fifth type.

Zydena enjoy rapid and predictable onset of action, duration of up to 24 hours, high in the class of PDE-5 inhibitors, the safety profile, Zydena not have testicular toxicity. Certainly, all of these properties will be the best in its segment.

The composition and the form of Udenafil

Tablets, film-coated light-pink color with light-yellow shade, oval shaped, imprinted with the symbol “100” on one side and symbols in the form of risk sharing letters “Z” and “Y” – to another, on a break – a white or nearly white .

1 tablet contains 100 mg udenafil;

excipients:

  • lactose
  • maize starch
  • colloidal silicon dioxide
  • L-hydroxypropylcellulose
  • hydroxypropyl-LF
  • talc
  • magnesium stearate.

1 or 4 tablets per pack.

Pharmacological action of Udenafil

Zydena – a drug for treatment of erectile dysfunction. Is a reversible selective inhibitor of cGMP-specific phosphodiesterase type 5 (PDE5).

Udenafil no direct relaxing effect on isolated corpus cavernosum, but enhances sexual stimulation relaxing effect of nitric oxide by inhibiting PDE-5, responsible for the breakdown of cGMP in the cavernous body. The result is relaxation of smooth muscles of arteries and blood flow to the tissues of the penis that causes erections. The drug has no effect in the absence of sexual stimulation.

Zydena improves erection and the possibility of successful sexual intercourse. The action of the drug has an optimal duration – up to 24 h. The effect is manifested as early as 30 minutes after taking the drug in the presence of sexual arousal.

In the study udenafil, men revealed no clinically significant effect on the drug quantity and concentration of sperm motility and morphology of spermatozoa.

Udenafil Indications

Treatment of erection disorders, characterized by the inability to achieve or maintain penile erection sufficient for satisfactory sexual intercourse.

Udenafil Dosing and Administration

Pills taken by mouth, with or without food, for 30 minutes before the alleged sexual activity.

Recommended dose – 100 mg. If necessary, taking into account individual performance and portability, the dose may be increased to 200 mg. The maximum recommended frequency of application – 1 times / day.

Udenafil Side effects

  • flushing
  • dizziness, eye pain
  • increased lacrimation
  • nasal congestion
  • headache

Also noted: palpitations, prolonged erections.

Cautions

Sexual activity is a potential risk for patients with cardiovascular disease, hypertension, so treatment of sexual dysfunctions, including use of Zydena, should not hold for men with heart disease, in which sexual activity is not recommended.

Patients with obstruction of blood outflow from the left ventricle (aortic stenosis) may be more sensitive to the action of vasodilators, including inhibitors of PDE. Despite the lack of clinical trials of cases of prolonged erection (longer than 4 hours) and priapism (painful erection lasting more than 6 h), such phenomena are peculiar to this class of drugs. In the event of an erection lasting more than 4 hours (regardless of pain), patients should immediately seek medical help. In the absence of timely treatment of priapism can lead to irreversible damage to the erectile tissue and erectile function.

In the absence of clinical data on the use udenafil in patients older than 71 y.o. this category not recommended for patients taking the drug. Not recommended for use Zydena in combination with other treatments for erectile dysfunction.

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  • rapid and predictable onset of action
  • provides necessary to erection hardness
  • increases the axial load on the penis
  • reduces the time of the refractory period (time after ejaculation until the next erection)
  • optimal duration of up to 24 hours
  • high safety profile in the class of PDE-5 inhibitors
  • Drinking alcohol and fatty food does not affect the action of udenafil
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Xenical

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84 Caps x 120mg Total 10080mg

Xenical (Orlistat)

Using Directions

The drug is prescribed for the frankly obese and for merely overweight people who have other health problems such as high blood pressure, diabetes, or high cholesterol levels. Your weight status is determined by your body mass index (BMI), a comparison of height to weight.

Along with dietary fat, Xenical decreases the absorption of some fat-soluble vitamins and beta-carotene. To compensate, you should take a multivitamin containing vitamins A, E, D, and K once a day, at least 2 hours before or 2 hours after taking Xenical

Do not take Xenical if you suffer from "chronic malabsorption syndrome"—a condition that prevents nutrients from passing from your stomach into your bloodstream—or from cholestasis, a blockage in the supply of bile needed for digestion. You’ll also need to avoid Xenical if it gives you an allergic reaction.

Take a capsule of Xenical during, or up to 1 hour after, each main meal. You should follow a nutritionally balanced, low-calorie diet that provides no more than 30 percent of its calories from fat. If you miss a meal, or the meal contains no fat, you can skip the accompanying dose of Xenical.

If you miss a dose, resume taking Xenical at the next meal. Don”t try to make up the loss with a double dose. The extra drug won”t help.

Store at room temperature, in a tightly sealed container.

Cautions

Weight loss begins within 2 weeks and continues for 6 to 12 months. The effect of using Xenical for more than 2 years is still unknown.

Side effects such as diarrhea and abdominal pain may be worse if you continue eating a high fat diet or even take a high-fat meal. Limit your fat intake.

Your doctor will test your thyroid function before starting you on Xenical to make sure that your weight problem is not due to an underactive thyroid gland (hypothyroidism). Xenical is not an appropriate remedy for this problem.

Xenical increases the likelihood of kidney stones. Use it with caution if you have a history of this problem.

If you have diabetes, weight-loss is likely to reduce your blood sugar levels. If you”re taking an oral diabetes medication or insulin, your dose may have to be reduced.

Note that the safety and efficacy of this drug in children have not been established.

Possible Side Effects

Side effects of Xenical are more common during the first year of treatment. If any develop or change in intensity, inform your doctor as soon as possible. Only your doctor can determine if it is safe for you to continue taking Xenical.

More common side effects may include: Abdominal discomfort or pain, anxiety, arthritis, back pain, diarrhea, dizziness, earache, fatigue, fatty or oily stools, fecal urgency or incontinence, flu, gas with fecal discharge, gum problems, headache, increased defecation, menstrual problems, muscle pain, nausea, oily discharge, rectal discomfort or pain, respiratory tract infections, skin rash, sleep problems, tooth problems, urinary tract infections, vaginal inflammation, vomiting

Less common side effects may include: Dry skin, ear/nose/throat problems, joint disorders

Side effects that usually occur after the first year of treatment with Xenical include: depression, leg pain, swollen feet, and tendonitis.

Possible food and drug interactions

If Xenical is taken with certain other drugs, the effects of either could be increased, decreased, or altered. It is especially important to check with your doctor before combining Xenical with the following:

Cyclosporine (Neoral and Sandimmune)

Pravastatin (Pravachol)

Warfarin (Coumadin)

The effects of Xenical during pregnancy have not been adequately studied and the drug is not recommended for pregnant women. If you are pregnant or plan to become pregnant, inform your doctor immediately.

It is not known whether Xenical appears in breast milk. Do not take it while breastfeeding

Dosage instructions

For adults recommended dose is one 120-milligram capsule 3 times daily with each main meal containing fat.

The results of a massive overdose of Xenical are unknown, although the drug seems relatively harmless. However, any medication taken in excess can have serious consequences. If you suspect an overdose, seek medical attention.

XenicalTM is a registered trademark of F. Hoffmann-La Roche Ltd

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Winstrol Oral

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100 Tabs x 10mg Total 1000mg

Winstrol tabs [Stanabol] (Stanozolol, Stromba)

Oral Winstrol

Oral Winstrol is an Oral version of Winstrol Depot (Stanozolol). So read all information about this product as for injectable form.

As it has been already mentioned, injectable version is more efficient than the winstrol oral one but this is mostly because oral Winstrol is used in lower dosages than injectable one and athletes simply don’t receive enough substance. If you take 50 mg of oral Winstrol a day, the results will be almost par with 50 mg of Winstrol depot, however, you may have problems with stomach and liver.

From the other hand, oral Winstrol is a good gear for females, they can do just 5-10 mg/ED and thus negative effects described above will not occur. Furthermore, oral Winstrol allows splitting daily dosage on two equal parts.

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Winstrol Depot

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Centrino Laboratories (Thailand)
5 Vials x 10ml. [50mg./ml.] Total 2500mg
CS Balkan Pharmaceuticals (Moldova)
15 Amps x 1ml. [50mg./ml.] Total 750mg
Balkan Pharmaceuticals (Moldova)
100 Tabs x 10mg Total 1000mg

Winstrol Depot (StanoJect, Stanozolol, Stanabol, Stromba, StrombaJect)

Winstrol (Winstrol Depot, oral Winstrol) is a brand name of very popular anabolic steroid called Stanozolol, which is a derivative of DHT (dihydrotestosterone). It has low androgenic ratio and thus low possibility of aromatization and estrogen-related side effects.

It’s primarily usage in bodybuilding is cutting (relief) Tables of Cycles. However, Winstrol is widely used not only by bodybuilders but also by non-bodybuilding athletes such as runners, cyclists, football players, soccer or hockey players and fighters of all kinds (kick-boxers for instance); i.e. in the sports where you have to be swift but not too heavy, because it provides you with lean mass and improves your strength without gaining excessive muscles.<

Stanozolol is one of the chemicals, which allowed amazing results to famous runner and simply exceptional athlete Ben Johnson. This substance provided him with a noticeable gain in muscle mass and relief, which could be perfect even for professional bodybuilder.

So, Winstrol is a very effective steroid when used properly. It is important to distinguish between two forms of Winstrol-Stanozolol, first is long-acting injectable version called Winstrol depot. Second is short-acting oral one (Winstrol oral). Winstrol depot is more effective and thus preferred by most athletes.

The main usage of Winstrol (Winstrol Depot) in bodybuilding is preparation for a competition. When complemented by a proper calorie-rich and protein-rich diet, Winstrol Depot provides the muscles with firmness and elasticity. Unfortunately, due to its low androgenic component, it is unable to protect the athlete from damages to muscle tissue. The absence of androgenic effect is compensated by stacking with Parabolan. The combination of injectable Winstrol 50 mg per day and Parabolan 2-3 amps / week is "a combination of top championships".<

Winstrol is good not only for preparation for a competition, but also in the bulking phase. Due to low water retention rapid weight gains with Winstrol are unlikely to occur. It provides rather moderate amount of lean and dry mass, which preserves after the cycle is over.

Injections of Winstrol in certain muscle groups are gaining in popularity because athletes have noticed that this leads to an accelerated growth of the affected muscles.

Dosage and usage

Injectable version is just slightly more efficient than the oral one and it’s not being destroyed by the liver. Because of this oral Winstrol requires a little bit higher dosages, however, most of athletes underdose it due to gastrointestinal pain and increased liver values – oral Winstrol is liver-toxic. So, here is where the myth of superiority of injectable Winstrol comes from. People simply can’t take equal dosages of oral version. Common dosage of oral Stanozolol is 15-30 mg/ED, daily dosage should be split on two parts – in the morning and evening during a meal, drink a liquid along with it.

Feature of the injectable Winstrol Depot is that its substance is dissolved in the water and not oil unlike most of other steroids. Therefore, intervals between injections with Winstrol Depot must be shorter comparing to other oil-based steroids like Primobolan, Deca-Duraboline, SuStanon, Parabolan, etc. because its lifetime is much shorter. Practice has shown that Winstrol Depot should be administered at least twice a day and the best results are observed at a daily dose of 50mg. (300-350 mg/week). Milder dosage is 50 mg/EOD (150 mg/week)

Inject deep in muscles and constantly rotate the spots. However, if athlete wants to promote particular muscle group injections should be done into it.

Winstrol Stacking

Winstrol (Stanozolol) is all-purpose steroid, however, we should admit that in first turn it’s a cutting agent for bodybuilder and it plays rather limited role in bulking cycles. The main reason for using it in non-cutting cycles is that in limited dose it can lower SHBG, which, in turn, increases the amount of free testosterone in the body
Depending on the level of the athlete, one usually takes 50 mg of long-acting Winstrol /ED or EOD and Parabolan 76 mg/ every 1 – 3 days. Although there is no scientific evidence in favor of special interaction between Winstrol Depot and Parabolan, it’s very likely that a synergistic effect appears basing on real-world evidence. Other steroids that well stack with Winstrol during pre-competition (cutting) cycle are Masterolone, Boldenone, Halotestin, Oxandrolone (anavar), Testosterone propionate, Primobolan and human growth hormone (:HGH

Bodybuilders who want to build up strength and mass often combine Winstrol injectable with Dianabol, Anadrol 50 (Anapolon, Oxymetholone), Testosterone,(long-acting) and Deca-Durabolin. With the combination of Anadrol 50 100 mg/ED, 50 mg Winstrol depot 50 mg/ED and 400 mg of Deca / week athlete is slowly coming to the ambitious results.

Aged athletes and steroid novices can achieve good progress with Winstrol depot and Deca-Durabolin or Winstrol depot and Primobolan

Cycle 0:

Winstrol depot 50 mg/ED is a cutting stack. Some people may do 50 mg/ED, it’s more aggressive.

Cycle 1:

Winstrol 100-150 mf/week + Primobolan Depot (Methenolone Enanthate) 200-300 mg/week for 6 weeks as a cutting phase AFTER regular deca-dianabol cycle

Cycle 2

Oxandrolone (anavar) 20-30 mg/ED + Winstrol 150 mg/week + clenbuterol 120 mg/ED for 12 weeks;
prabolan 152-228 mg/week for the first 8 weeks; Proviron (Masterlone) 300 mg/week + Cytomel T3 increase from 25 to 100 mg / week during weeks 9-12

Cycle 3

Winstrol 150 mg/w + Parabolan Depot 152 mg/w

Cycle 4

Winstrol (150 mg/w) + Dianabol (20-30 mg/ED) + Testosterone Propionate (150 mg/w) for 8-10 weeks + Clenbuterol at the end

Cycle 5

Winstrol 50-100 mg/w + Deca-Durabolin 300-200 mg/w

Cycle 6

Winstrol oral 40-60mg/ED + Boldabol (Equipoise) 100-200 mg/w

Cycle 7

Winstrol + Trenbolone + Clenbuterol – relief cycle for novices.

Cycle 8

Primobolan Depot (Methenolone Enanthate) 200-300 mg/w + Winstrol 150-300 mg/w + Anavar (Oxandrolone) 20-60 mg/ED + Clenbuterol + PCT (Tamoxifen (Nolvadex) and HCG) – relief for advanced users

Cycle 9

Boldenone Undecylenate 300 mg/w + Winstrol oral 40 mg/ED + Nandrolone Decanoate (Phenilpropionate) 300 mg / w – relief for advanced users

Detection time

Oral Stanozolol – 3 weeks

Injectable Stanozolol (Winstrol depot) – 3 months

Side effects and PCT (Post Cycle Therapy) with Winstrol

Only small number of athletes report water retention or other negative effects. However, one should be aware that oral Winstrol can be toxic to the liver in excessive dosages.

Other non-androgenic side effects, which might occur are: headaches, muscle spasms, in rare cases high blood pressure can occur. The possibility of liver damage in the form of injectable Winstrol is very small, but still in high doses may increase the liver values.

Because the Winstrol Depot is dissolved in the water, injection, in common is more painful comparing to oil-based gear and have to be taken more frequently. This leads to another negative effect – scar tissue on the often injection spots, which cause athletes t inject not only into buttocks but also to shoulders, legs or even calves. Athletes wishing to avoid this take Winstrol Depot twice a week for 2-3ml. This decreases effectiveness but decreases pain and prevents scar tissue appearance.

As with most of other steroids, Winstrol suppresses natural hormonal levels although not to that extension as many others. Running testosterone in a cycle containing Winstrol helps to avoid possible sexual dysfunction.
After Winstrol cycle is over it’s necessary to do PCT: First week: 40mg of tamoxifen or 100mg clomiphen/ED or combo of both. One-two more weeks: 20mg of tamoxifen or 50mg clomiphen or combo of both.

Female usage

It’s one of the few substances, which could be used more or less safely by females in low dosages because it has more anabolic properties than androgenic ones. But occasionally Winstrol can cause virilization, even this small androgenic component may, become noticeable for women with a dose of only 50 mg per week. And troubles are almost guaranteed for female athletes with a dosage of 100 mg / week. Despite Winstrol moves out quickly, it can cause undesired accumulation of androgens in the female body, which cause virilization effects such as deep voice, hair growth, hypersexuality, etc. (something similar happens to some of natural brunettes). However, ambitious female athletes still use it 50 mg / EOD disregarding all side effects.
Normally, female athlete can tolerate around 5-10mg of Stanosolol per day, which perfectly fits for oral Winstrol usage

Winstrol fakes

Due to popularity of Winstrol there are many fakes on the market. The first thing to mention is that British Dragon Winstrol depot and Stanozolol (oral Winstrol) is no longer manufactured since they got busted, It might be still in circulation till the end of 2011 but anything with manufacture date after 2008 is a fake.

Brief description of Stanozolol:

Activity: 48 hours
Classification: Anabolic / Androgenic Steroid
Dose: Men 25-100 mg / day
Acne: Rare
Water Retention: Rare
High Blood Pressure: Rare
Hepatotoxicity: Yes, it is 17-Alpha alkalized
Aromatization: No, it is a derivative of DHT
DHT Conversion: No
Decrease HPTA function: Weak

Advantages

There are several reliable sources where you can buy anabolic steroids: